White Or Yellow Powder Mibolerone CAS 3704-09-04 Muscle Growth Hormone , Oral Anabolic Steroid

Mibolerone

Cas number : 3704-09-04
Chemical Formula: C20-H30-O2
Molecular Weight: 302.455
Description: white or yellow white crystalline powder

Mibolerone is a synthetic anabolic steroid. It binds both androgen and progesterone receptors and exerts both androgenic and progestagenic actions. Mibolerone (CHEQUE® Drops) was used in veterinary for estrous (heat) prevention in adult female dogs not intended primarily for breeding purposes. No prescription preparation, human or veterinary, is currently known to contain mibolerone worldwide.

 

 

General description

The synthetic androgen mibolerone (7α,17α dimethyl-19-nortestosterone) is an androgenic steroid.

Biochem/physiol Actions

The synthetic androgen mibolerone (7α,17α dimethyl-19-nortestosterone) reversibly blocks the multiplication of LNCaP (human prostate carcinoma cell line) cells. In prostate, liver, and cultured cells, it serves as an efficient radioactive ligand for the quantitation and characterization of androgen receptors.

Mibolerone is a synthetic anabolic steroid with a similar profile of activity as R1881 (Metribolone) with a higher affinity (Kd = 1.5 nM) for the androgen receptor in human prostate tissue than R1881 (Kd = 2.3 nM).

 

Activation of androgen receptor in epidermal growth factor modulation of fetal mouse sexual differentiation.

1996 Oct 14

8912815

Expression of the human androgen receptor in eukaryotic cells using a recombinant adenovirus vector yields high levels of the soluble, functional receptor protein.

2001 Dec

11719284

Characterization of intracellular aggregates using fluorescently-tagged polyglutamine-expanded androgen receptor.

2001 Jul

15111251

Regulation of u-PA gene expression in human prostate cancer.

2001 Nov 1

11745419

Melatonin elicits nuclear exclusion of the human androgen receptor and attenuates its activity.

2001 Oct 1

11582594

 

 

 

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